PD 123319 ditrifluoroacetate

CAS No. 136676-91-0

PD 123319 ditrifluoroacetate( PD123319 ditrifluoroacetate | PD-123319 ditrifluoroacetate )

Catalog No. M11516 CAS No. 136676-91-0

A potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    PD 123319 ditrifluoroacetate
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.
  • Description
    A potent, selective, non-peptide AT2 receptor with IC50 of 34 nM.Heart Failure Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    PD123319 ditrifluoroacetate | PD-123319 ditrifluoroacetate
  • Pathway
    GPCR/G Protein
  • Target
    Angiotensin Receptor
  • Recptor
    Angiotensin Receptor
  • Research Area
    Cardiovascular Disease
  • Indication
    ——

Chemical Information

  • CAS Number
    136676-91-0
  • Formula Weight
    736.6575
  • Molecular Formula
    C35H34F6N4O7
  • Purity
    >98% (HPLC)
  • Solubility
    H2O: ≥ 36 mg/mL
  • SMILES
    CC1=C(C=CC(=C1)CN2C=NC3=C2CC(N(C3)C(=O)C(C4=CC=CC=C4)C5=CC=CC=C5)C(=O)O)N(C)C.C(=O)(C(F)(F)F)O.C(=O)(C(F)(F)F)O
  • Chemical Name
    1H-Imidazo[4,5-c]pyridine-6-carboxylic acid, 1-[[4-(dimethylamino)-3-methylphenyl]methyl]-5-(2,2-diphenylacetyl)-4,5,6,7-tetrahydro-, (6S)-, 2,2,2-trifluoroacetate (1:2)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Blankley CJ, et al. J Med Chem. 1991 Nov;34(11):3248-60. 2. Keiser JA, et al. J Pharmacol Exp Ther. 1992 Sep;262(3):1154-60. 3. Macari D, et al. Eur J Pharmacol. 1993 Nov 2;249(1):85-93.
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